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Signaling Pathways - COX - Calcium chelator - Ubiquitin-specific proteases - Cytochrome P450 (CYP450)

31件产品中的 21-30

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  1. Posaconazole
    A1718 Posaconazole
    中文名: 泊沙康唑
    Target: Cytochrome P450 (CYP450)|sterol demethylase
    Summary: 甾醇 C14ɑ去甲基化酶抑制剂
      ≥35.04 mg/mL
      insoluble in H2O
  2. Celecoxib
    A1664 Celecoxib
    中文名: 塞来昔布
    Target: COX
    Summary: COX-2选择性抑制剂
      ≥19.07 mg/mL
      insoluble in H2O
  3. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  4. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  5. Bardoxolone
    A3220 Bardoxolone
    中文名: 巴多索隆
    Target: COX|iNOS
    Summary: 用于治疗慢性肾病,每天一次
      ≥49.2 mg/mL
      insoluble in H2O
  6. Clarithromycin
    A4322 Clarithromycin
    中文名: 克拉霉素
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A抑制剂
      ≥31.2 mg/mL
      insoluble in H2O
  7. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  8. Cobicistat (GS-9350)
    A4313 Cobicistat (GS-9350)
    中文名: 可比司他
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A的选择性抑制剂
      ≥150.9 mg/mL
      insoluble in H2O
  9. Abiraterone acetate
    A8202 Abiraterone acetate
    中文名: 乙酸阿比特龙酯
    Target: Cytochrome P450 (CYP450)
    Summary: 细胞色素p450 17a1抑制剂
      ≥11.22 mg/mL
      insoluble in H2O
  10. Resveratrol
    A4182 Resveratrol
     2 Citation
    中文名: 白藜芦醇
    Target: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductase
    Summary: SIRT1激活剂
      ≥9.65 mg/mL
      insoluble in H2O

31件产品中的 21-30

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