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Signaling Pathways - Smoothened - Bromodomain and Extra-Terminal motif (BET) - Histamine H1 Receptors - S1P receptors

21件产品中的 11-20

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  1. PF-04449913
    B3283 PF-04449913
    中文名: 格拉吉布
    Target: Smoothened
    Summary: Smoothened拮抗剂
      ≥20.15 mg/mL
      insoluble in H2O
  2. BAF312 (Siponimod)
    B3225 BAF312 (Siponimod)
     1 Citation
    中文名: 辛波莫德
    Target: S1P receptors
    Summary: S1P受体激动剂
      ≥194.8 mg/mL
      insoluble in H2O
  3. Fingolimod (FTY720)
    A8548 Fingolimod (FTY720)
    中文名: 盐酸芬戈莫德
    Target: S1P receptors
    Summary: S1P受体激动剂
      ≥17.2 mg/mL
      ≥31.3 mg/mL
  4. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  5. Paliperidone
    A8496 Paliperidone
    中文名: 帕利哌酮
    Target: 5-HT2 Receptors|D2 Receptors|D3 Receptors|5-HT1 Receptors|Histamine H1 Receptors
    Summary: 多巴胺受体拮抗剂
      ≥10.662 mg/mL
      insoluble in H2O
  6. Cyclopamine
    A8340 Cyclopamine
     1 Citation
    中文名: 环巴胺
    Target: Smoothened
    Summary: Hedgehog (Hh)信号抑制剂
      ≥6.86 mg/mL
      insoluble in H2O
  7. Loratadine
    A2960 Loratadine
    中文名: 氯雷他定
    Target: Histamine H1 Receptors
    Summary: 外周HH1R拮抗剂
      ≥19.14 mg/mL
      insoluble in H2O
  8. Lidocaine
    A1450 Lidocaine
    中文名: 利多卡因
    Target: Histamine H1 Receptors
    Summary: 麻醉剂和Ib类抗心律失常药
      ≥11.72 mg/mL
      insoluble in H2O
  9. LDE225 Diphosphate
    A3543 LDE225 Diphosphate
    Target: Smoothened
    Summary: Smo拮抗剂
      ≥27.85 mg/mL
      insoluble in H2O
  10. Clemizole hydrochloride
    A3316 Clemizole hydrochloride
    中文名: 盐酸克立咪唑
    Target: Histamine H1 Receptors|TRPC channel
    Summary: H1组胺受体拮抗剂
      ≥18.12 mg/mL
      ≥5.12 mg/mL

21件产品中的 11-20

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