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- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂
- B6011 A-12104772 CitationTarget: Mcl-1Summary: MCL-1抑制剂
- A3517 JDTicSummary: 阿片受体拮抗剂
- A3723 Phloretin中文名: 根皮素Target: SGLTSummary: 在苹果中发现的二氢查耳酮
- A1907 5-Azacytidine6 Citation中文名: 氮胞苷(5-氮胞苷)Target: DNA MethyltransferasesSummary: DNA甲基转移酶抑制剂
- A8403 CP-91149Target: Glycogen PhosphorylasesSummary: 糖原磷酸化酶选择性抑制剂
- A4093 ITF2357 (Givinostat)2 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC抑制剂
- A4061 IPI-504 (Retaspimycin hydrochloride)3 Citation中文名: 瑞他霉素盐酸盐Target: HSP90Summary: Hsp90抑制剂
- A8650 Saxagliptin中文名: 沙格列汀Target: DPP-4Summary: DPP4抑制剂
- B1879 AdipoRonTarget: AdipoR1|AdipoR2Summary: AdipoR1/2激动剂