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- B5851 FG2216Target: Pyruvate dehydrogenases (PDH)Summary: HIF-脯氨酰羟化酶抑制剂
- B2157 Cabazitaxel3 Citation中文名: 卡巴他赛Target: Microtubule/TubulinSummary: 微管相关抑制剂
- A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH抑制剂
- A3394 Epothilone D中文名: 埃博霉素 DTarget: Microtubule/TubulinSummary: 天然聚酮化合物
- A1765 Vincristine sulfate中文名: 硫酸长春新碱Target: Microtubule/TubulinSummary: 微管的破坏者,抗肿瘤剂
- A8601 Tankyrase Inhibitors (TNKS) 49Target: TankyrasesSummary: 端锚聚合酶抑制剂