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- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- A2249 T0901317Target: Liver X receptors (LXRs)Summary: 肝X受体激动剂
- B1054 Resiquimod (R-848)2 Citation中文名: 雷西莫特,瑞喹莫德Target: Toll-like receptors (TLRs)Summary: 免疫应答调节剂
- B7336 Thiostrepton中文名: 硫链丝菌素Target: FoxM1Summary: 抑制细菌蛋白合成的抗生素
- B5551 Poly(I:C)Target: Toll-like receptors (TLRs)Summary: Toll样受体3(TLR3)激动剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂