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- A1832 Doxorubicin (Adriamycin) HCl2 Citation中文名: 盐酸多柔比星,盐酸阿霉素Target: TopoisomerasesSummary: 抗肿瘤抗生素,抑制TOPO II。
- A4536 Fostriecin sodium saltTarget: PP1|PP2A|Topoisomerases|PP4Summary: 抗肿瘤抗生素
- B6274 N-AcetyltryptamineTarget: Melatonin ReceptorsSummary: 褪黑激素受体调节剂
- B7426 L189Target: DNA LigasesSummary: DNA连接酶 I、III 及IV的抑制剂
- B7382 Ellipticine中文名: 玫瑰树碱,椭圆玫瑰树碱Target: TopoisomerasesSummary: DNA拓扑异构酶II抑制剂
- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- A1748 Ramelteon1 Citation中文名: 雷美替胺Target: Melatonin ReceptorsSummary: MT1/MT2激动剂