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- A4356 Varespladib (LY315920)中文名: 伐瑞拉迪Target: PhospholipasesSummary: HnsPLA的强效选择性抑制剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A8476 MK-2461Target: FLT3|PDGFR|MET|RonSummary: C-Met(野生型/突变型)抑制剂
- B2087 Ciclopirox中文名: 环吡酮胺Target: HydroxylasesSummary: 广谱抗真菌剂
- B1823 Quinacrine 2HCl中文名: 盐酸奎纳克林Target: Phospholipases|Monoamine oxidases (MAOs)Summary: 抗原虫剂
- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂