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- A8328 LDK378中文名: 色瑞替尼Target: ALKSummary: 强效的ALK抑制剂
- B6304 Etazolate hydrochloride2 CitationTarget: Phosphodiesterases (PDEs)Summary: PDE-4抑制剂和选择性GABA-A受体调节剂
- A3196 AT-101中文名: (R)-(-)-棉子酚Target: NS3/4a ProteasesSummary: BH3-类似物,棉酚对映异构体
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂