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- A2487 Odanacatib (MK-0822)中文名: 奥当卡替Target: CathepsinsSummary: 组织蛋白酶K抑制剂
- N2408 Genipin中文名: 京尼平Target: UCPSummary: 用于治疗2型糖尿病症状
- B7382 Ellipticine中文名: 玫瑰树碱,椭圆玫瑰树碱Target: TopoisomerasesSummary: DNA拓扑异构酶II抑制剂
- A4412 MDL 28170Target: Cathepsins|CalpainsSummary: Calpain和cathepsin B抑制剂
- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- A2576 E-642 CitationTarget: Cathepsins|Calpains|PapainsSummary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
- A2602 Calpain Inhibitor I, ALLN2 CitationTarget: Cathepsins|CalpainsSummary: Calpain I/II/ B/L抑制剂