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- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- A3967 Lapatinib Ditosylate中文名: 二苯磺酸拉帕替尼Target: EGFR|ErbB-2Summary: EGFR / HER2抑制剂
- B2082 Camostat Mesilate中文名: 甲磺酸卡莫司他Target: Trypsin-like proteaseSummary: 胰蛋白酶样蛋白酶抑制剂
- A3720 PF-83801 CitationTarget: AutotaxinSummary: Autotaxin抑制剂