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- A8324 LDN-193189Target: BMP and Other Activin ReceptorsSummary: ALK抑制剂
- A4024 Danoprevir (RG7227)中文名: 丹诺瑞韦Target: HCV ProteasesSummary: HCV NS3/4A蛋白酶抑制剂
- B3688 ML347Target: BMP and Other Activin ReceptorsSummary: 有效的BMP受体选择性抑制剂
- A4182 Resveratrol2 Citation中文名: 白藜芦醇Target: Sir2-like Family Deacetylases (Sirtuins)|COX|LOX|Adenylyl cyclase|Quinone reductaseSummary: SIRT1激活剂
- B1382 Anastrozole中文名: 阿那曲唑Target: AromatasesSummary: 芳香酶抑制剂
- A1307 Letrozole中文名: 来曲唑Target: AromatasesSummary: 非甾体类芳香酶抑制剂。