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- A1020 GnRH Associated Peptide (1-13), humanTarget: prolactin secretion|gonadotropin releaseSummary: 催乳素分泌抑制剂
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- B2136 Zanamivir中文名: 扎那米韦Target: Influenza virusesSummary: 流感A/B病毒神经氨酸酶抑制剂