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- A3967 Lapatinib Ditosylate中文名: 二苯磺酸拉帕替尼Target: EGFR|ErbB-2Summary: EGFR / HER2抑制剂
- A4509 PX 12Target: TrxSummary: Trx-1抑制剂
- B2082 Camostat Mesilate中文名: 甲磺酸卡莫司他Target: Trypsin-like proteaseSummary: 胰蛋白酶样蛋白酶抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂