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- B6552 CGP 20712 dihydrochlorideTarget: adrenoceptorSummary: β1拮抗剂
- B2160 LY2608204Target: GKSummary: GK激活剂
- N2172 5,7-dihydroxychromone1 Citation中文名: 5,7-二羟基色酮Target: Nrf2/ARE signal|PPARSummary: Nrf2/ARE信号激活剂和PPARγ激动剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A8474 Mirabegron (YM178)中文名: 米拉贝隆Target: adrenoceptorSummary: 选择性β3肾上腺素受体激动剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂