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- A1932 (-)-Huperzine A中文名: 石杉碱甲Target: NMDA Receptors|AChESummary: NMDA受体拮抗剂/AChE抑制剂
- A4181 EX 527 (SEN0014196)1 CitationTarget: SirtuinSummary: SIRT1抑制剂
- B1890 AZ191Target: DYRKSummary: DYRK1B抑制剂
- B1952 ID-8Target: DYRKSummary: DYRK抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂
- B1602 Donepezil HCl中文名: 盐酸多奈哌齐Target: AChESummary: AChE抑制剂