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- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A8815 SM-1648 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: 抗癌药
- A8607 PPY ATarget: Abl kinasesSummary: Abl激酶抑制剂
- A4224 GDC-01522 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAP 拮抗剂
- A1655 GW25801 CitationTarget: CSF-1RSummary: CFMS激酶/CSF-1R抑制剂
- A3022 Pazopanib (GW-786034)中文名: 帕唑帕尼Target: CSF-1R|VEGFR|PDGFR|c-Kit|FGFRSummary: (GW-786034)VEGFR/PDGFR/FGFR 的抑制剂。