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- A1036 Thrombin Receptor Activator for Peptide 5 (TRAP-5)Target: Thrombin ReceptorSummary: Thrombin Receptor Activator for Peptide 5
- A2574 Aprotinin1 Citation中文名: 抑酶肽Target: Trypsin|Chymotrypsin|Kallikrein|TrypsinogenSummary: 牛胰蛋白酶抑制剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- A4375 Anacetrapib (MK-0859)1 Citation中文名: 安塞曲匹Target: CETPSummary: RhCETP/突变型 CETP(C13S) 抑制剂
- A4377 Evacetrapib (LY2484595)Target: CETPSummary: 强效的CETP选择性抑制剂