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- A4071 Fluorouracil (Adrucil)3 Citation中文名: 氟尿嘧啶Target: Thymidylate SynthaseSummary: 胸苷酸合成酶抑制剂,抗肿瘤药物。
- B1685 Broxyquinoline中文名: 溴羟喹啉Target: Tetrahydrofolate dehydrogenaseSummary: 抗原虫剂
- A8711 DDD1074982 CitationTarget: Eukaryotic elongation factorsSummary: 新型的多级抗疟疾制剂
- B7675 DIDSTarget: voltage-gated chloride channelsSummary: 阴离子运输抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂