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- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- B7795 Toyocamycin中文名: 丰加霉素Target: phosphatidylinositol kinaseSummary: 腺苷类似物,抗肿瘤抗生素
- A4031 Telaprevir (VX-950)中文名: 特拉匹韦Target: HCV NS3-4A proteaseSummary: HCV NS3-4A蛋白酶抑制剂
- A8339 TAK-875Target: GPR40Summary: GPR40激动剂