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- A4216 Thalidomide中文名: 沙利度胺Target: Ubiquitin E3 LigasesSummary: 免疫调节剂,镇静药,血管生成抑制剂
- A4228 Nutlin-3Target: MDM2Summary: MDM2 拮抗剂
- B7795 Toyocamycin中文名: 丰加霉素Target: phosphatidylinositol kinaseSummary: 腺苷类似物,抗肿瘤抗生素
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂
- A3762 RG71125 CitationTarget: MDM2Summary: MDM2抑制剂