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- A4443 Gliotoxin1 CitationTarget: 20S proteasomal chymotrypsin|Geranylgeranyltransferase I|FarnesyltransferaseSummary: 20S蛋白酶体抑制剂
- A8432 Fenticonazole Nitrate中文名: 硝酸芬替康唑Target: Cytochrome P450 (CYP450)|Synthases/SynthetasesSummary: 抗真菌药
- A5588 Oligomycin A1 Citation中文名: 寡霉素ATarget: Synthases/SynthetasesSummary: 线粒体ATP合成酶抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A2278 NVP-AEW541Target: Insulin ReceptorSummary: IGF-IR抑制剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂