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- A4071 Fluorouracil (Adrucil)3 Citation中文名: 氟尿嘧啶Target: Thymidylate SynthaseSummary: 胸苷酸合成酶抑制剂,抗肿瘤药物。
- A8533 Terbinafine中文名: 特比萘芬Target: Squalene epoxidasesSummary: 烯丙胺抗真菌剂
- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂
- B1528 XL335Target: Farnesoid X receptors (FXRs)Summary: FXR激动剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- B2047 Terbinafine HCl中文名: 盐酸特比萘芬Target: Squalene epoxidasesSummary: 有效的非竞争性角鲨烯环氧酶抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂