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- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- B1488 Pramipexole中文名: 普拉克索Target: D2 Receptors|D3 Receptors|D4 ReceptorsSummary: 多巴胺激动剂
- A3635 MRT67307 HClTarget: TBK1|MARK1|NUAK1Summary: SIK/TBK-1/IKKe抑制剂
- A3374 Dronedarone中文名: 决奈达隆Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4和2D6抑制剂
- B2094 Fluconazole中文名: 氟康唑Target: Cytochrome P450 (CYP450)Summary: 三唑抗真菌剂
- A4316 Ketoconazole中文名: 酮康唑Target: Cytochrome P450 (CYP450)Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
- A1718 Posaconazole中文名: 泊沙康唑Target: Cytochrome P450 (CYP450)|sterol demethylaseSummary: 甾醇 C14ɑ去甲基化酶抑制剂
- A8401 Clotrimazole2 Citation中文名: 克霉唑Target: Cytochrome P450 (CYP450)Summary: 抗真菌化合物
- A8496 Paliperidone中文名: 帕利哌酮Target: 5-HT2 Receptors|D2 Receptors|D3 Receptors|5-HT1 Receptors|Histamine H1 ReceptorsSummary: 多巴胺受体拮抗剂
- A4322 Clarithromycin中文名: 克拉霉素Target: Cytochrome P450 (CYP450)Summary: CYP3A抑制剂