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- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A2570 Leupeptin, Microbial中文名: 亮抑酶肽Target: Cathepsins|Calpains|TrypsinsSummary: 丝氨酸和半胱氨酸蛋白酶抑制剂
- B6552 CGP 20712 dihydrochlorideTarget: adrenoceptorSummary: β1拮抗剂
- A4443 Gliotoxin1 CitationTarget: 20S proteasomal chymotrypsin|Geranylgeranyltransferase I|FarnesyltransferaseSummary: 20S蛋白酶体抑制剂
- A8474 Mirabegron (YM178)中文名: 米拉贝隆Target: adrenoceptorSummary: 选择性β3肾上腺素受体激动剂