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- A3494 INCB3344Target: CCRSummary: CCR2趋化因子受体拮抗剂
- A4031 Telaprevir (VX-950)中文名: 特拉匹韦Target: HCV NS3-4A proteaseSummary: HCV NS3-4A蛋白酶抑制剂
- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A1352 Zoledronic Acid中文名: 唑来膦酸Target: Farnesyl Diphosphate SynthasesSummary: 含氮二磷酸盐