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- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A3965 BI 25361 CitationTarget: PLK|Bromodomain-containing proteins(BRDs)Summary: ATP竞争性的Plk1抑制剂
- B1175 PalovaroteneTarget: RARsSummary: 选择性视黄酸受体γ(RAR-γ)激动剂
- B4702 AGN 1943101 CitationTarget: RARsSummary: Pan-RAR拮抗剂
- A1267 Adapalene中文名: 阿达帕林Target: RARsSummary: RARβ和RARγ激动剂