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- A4351 PluriSIn #1 (NSC 14613)Target: Stearoyl-CoA 9-desaturase (SCD-1)Summary: SCD1抑制剂
- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- A8525 Sotrastaurin (AEB071)Target: PKCSummary: PKC抑制剂
- B1287 Ro 31-8220Target: PKCSummary: Pan-PKC抑制剂
- A8351 VX-809中文名: 鲁玛卡托Target: CFTRSummary: CFTR调节剂