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- A4351 PluriSIn #1 (NSC 14613)Target: Stearoyl-CoA 9-desaturase (SCD-1)Summary: SCD1抑制剂
- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR抑制剂
- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- B3341 Sotalol hydrochloride1 Citation中文名: 盐酸索他洛尔Target: Inward Rectifier Potassium (Kir) ChannelsSummary: β-肾上腺素能受体拮抗剂
- A8312 Torin 17 CitationTarget: mTORSummary: MTOR抑制剂
- B1296 Glibenclamide中文名: 格列本脲Target: Inward Rectifier Potassium (Kir) ChannelsSummary: 胰岛素生产调节剂
- A8351 VX-809中文名: 鲁玛卡托Target: CFTRSummary: CFTR调节剂