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- A8316 PD 0332991 (Palbociclib) HCl5 Citation中文名: 帕博西尼Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- A3570 LY2090314Target: GSK-3Summary: 有效的GSK-3抑制剂
- B1174 LGX818中文名: 康奈非尼Target: RafSummary: RAF抑制剂
- A4135 Tofacitinib (CP-690550) Citrate2 Citation中文名: 托法替尼Target: JAKSummary: JAK抑制剂
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A8177 PAC-11 CitationTarget: CaspasesSummary: 半胱天冬酶-3酶原激活剂