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- B1874 4μ8C2 CitationTarget: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1 Rnase抑制剂
- B3288 APY29Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α变构调节剂
- B8023 Cerdulatinib (PRT062070)Target: JAK|Syk|TYK2Summary: Syk/JAK抑制剂
- A4147 LY2784544Target: Aurora Kinases|FLT3|VEGFR|FGFR|Trk Receptors|JAK|ALK|TYK2|MUSK|MAP3KSummary: JAK2抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂