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- A1877 XAV-9391 CitationTarget: TNKSSummary: Tankyrase 1/2抑制剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- A8328 LDK378中文名: 色瑞替尼Target: ALKSummary: 强效的ALK抑制剂
- A3799 SB-505124 hydrochlorideTarget: ALKSummary: TGF-β/活化素信号传导中ALK5/ALK4/ALK7 的抑制剂