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- A8620 AZD-34633 CitationTarget: ALK|Insulin-like growth factors (IGFs)Summary: ALK/IGF1R抑制剂
- A3825 SLx-21191 CitationTarget: ROCKSummary: ROCK2抑制剂
- A5611 GSK429286ATarget: ROCKSummary: 选择性ROCK1/ROCK2抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂