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- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- A2402 Floxuridine中文名: 氟尿苷Target: Synthases/SynthetasesSummary: 抗肿瘤抗代谢物
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- B1472 Mizoribine中文名: 咪唑立宾Target: Synthases/SynthetasesSummary: DNA/RNA合成抑制剂