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- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8170 Z-FA-FMKTarget: cysteine proteaseSummary: 半胱氨酸蛋白酶抑制剂
- A4322 Clarithromycin中文名: 克拉霉素Target: Cytochrome P450 (CYP450)Summary: CYP3A抑制剂
- A8703 IsosafroleTarget: Lactate Dehydrogenases (LDH)Summary: stiripentol类似物,有效的LDH抑制剂。
- A8704 Stiripentol中文名: 司替戊醇Target: Lactate Dehydrogenases (LDH)Summary: LDH抑制剂
- B2094 Fluconazole中文名: 氟康唑Target: Cytochrome P450 (CYP450)Summary: 三唑抗真菌剂
- A8162 E-64-c中文名: 阿洛司他丁酸Target: cysteine proteaseSummary: 半胱氨酸蛋白酶抑制剂
- A8537 Thioridazine HCl中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 ReceptorsSummary: 钙通道蛋白抑制剂
- A4316 Ketoconazole中文名: 酮康唑Target: Cytochrome P450 (CYP450)Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
- A1718 Posaconazole中文名: 泊沙康唑Target: Cytochrome P450 (CYP450)|sterol demethylaseSummary: 甾醇 C14ɑ去甲基化酶抑制剂