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- A4351 PluriSIn #1 (NSC 14613)Target: Stearoyl-CoA 9-desaturase (SCD-1)Summary: SCD1抑制剂
- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- B2189 YM201636Target: PIKfyveSummary: PIKfyve抑制剂
- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂