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- A4393 Paclitaxel (Taxol)4 Citation中文名: 紫杉醇Target: Microtubules/TubulinsSummary: 抗肿瘤药
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- A1630 Epothilone B (EPO906, Patupilone)中文名: 埃博霉素B,帕土匹龙Target: Microtubules/TubulinsSummary: 大环内酯物抗癌试剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- A8487 Nocodazole1 Citation中文名: 诺考达唑Target: Microtubules/TubulinsSummary: 微管蛋白产生抑制剂,抗肿瘤剂
- A3183 Ansamitocin P-3中文名: 安丝菌素 P 3'Target: Microtubules/TubulinsSummary: 美登素类似物,微管蛋白抑制剂