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- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A4483 PRIMA-1Target: p53Summary: BAX抑制剂
- A3408 Exendin-4中文名: 艾塞那肽Target: Glucagon-like peptide 1 (GLP-1) receptorsSummary: GLP-1激活剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A1755 Tenofovir Disoproxil Fumarate中文名: 富马酸替诺福韦酯Target: Reverse TranscriptasesSummary: 抗逆转录制剂(HIV-1 RT 抑制剂)