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- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A8324 LDN-193189Target: BMP and Other Activin ReceptorsSummary: ALK抑制剂
- B3688 ML347Target: BMP and Other Activin ReceptorsSummary: 有效的BMP受体选择性抑制剂
- B1175 PalovaroteneTarget: RARsSummary: 选择性视黄酸受体γ(RAR-γ)激动剂
- B4702 AGN 1943101 CitationTarget: RARsSummary: Pan-RAR拮抗剂
- A1267 Adapalene中文名: 阿达帕林Target: RARsSummary: RARβ和RARγ激动剂