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- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A8189 PSI-62063 CitationTarget: HCV polymeraseSummary: HCV RNA聚合酶抑制剂
- A3358 DeltarasinTarget: Phosphodiesterases (PDEs)Summary: KRAS-PDEδ相互作用抑制剂
- B1386 Milrinone中文名: 米力农Target: Phosphodiesterases (PDEs)Summary: PDE3抑制剂
- A3738 PSI-7977中文名: 索非布韦,索氟布韦Target: HCV polymeraseSummary: 慢性丙型肝炎病毒(HCV)感染的抗病毒剂
- B6367 NPPBTarget: Calcium-activated chloride channels (CaCC)|GPR35Summary: 氯离子通道抑制剂
- A4032 VX-222 (VCH-222, Lomibuvir)Target: HCV polymeraseSummary: HCV RNA聚合酶抑制剂
- B1476 Raltitrexed中文名: 雷替曲塞Target: Thymidylate SynthaseSummary: 胸苷酸合酶抑制剂
- A4071 Fluorouracil (Adrucil)3 Citation中文名: 氟尿嘧啶Target: Thymidylate SynthaseSummary: 胸苷酸合成酶抑制剂,抗肿瘤药物。
- A4346 Aminophylline中文名: 氨茶碱,氨基非林Target: Phosphodiesterases (PDEs)Summary: Pan-PDE抑制剂