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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- B1374 WZ4003Target: NUAK1|NUAK2Summary: NUAK1/2抑制剂
- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B2068 Zafirlukast中文名: 扎鲁司特Target: Leukotriene and Related ReceptorsSummary: 口服白三烯受体拮抗剂
- B7023 MK-571Target: Leukotriene and Related ReceptorsSummary: leukotriene D4(LTD4)受体拮抗剂
- A3635 MRT67307 HClTarget: TBK1|MARK1|NUAK1Summary: SIK/TBK-1/IKKe抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂