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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- N1842 Taxifolin中文名: 紫杉叶素,黄杉素Target: AdipoR2|Opioid receptors
- B1211 AICAR phosphate中文名: 阿卡地新磷酸盐Target: AMPKSummary: AMPK激活剂
- A3317 Clozapine N-oxide(CNO)1 Citation中文名: 氯氮平的N-氧化物Target: DREADD LigandsSummary: Clozapine代谢产物,用于化学遗传学
- B1373 Phenformin HCl1 Citation中文名: 盐酸苯乙双胍,盐酸苯乙福明Target: AMPKSummary: 抗糖尿病
- B6020 GSK6211 CitationTarget: AMPKSummary: AMPK激动剂
- B3252 Dorsomorphin (Compound C)5 CitationTarget: AMPKSummary: AMPK抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂