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- B1518 Erteberel (LY500307)Target: Estrogen and Related ReceptorsSummary: ERβ激动剂
- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A8425 Estradiol中文名: 雌二醇Target: Estrogen and Related ReceptorsSummary: 性激素
- B5961 Cytosporone BTarget: Nur77Summary: 核孤儿受体Nur77的激动剂
- B1111 N6022Target: S-nitrosoglutathione reductaseSummary: GSNOR抑制剂
- B1506 Estradiol valerate中文名: 戊酸雌二醇Target: Estrogen and Related ReceptorsSummary: 雌激素受体激动剂
- B1513 Toremifene Citrate中文名: 枸橼酸托瑞米芬Target: Estrogen and Related ReceptorsSummary: 口服选择性雌激素受体调节剂(SERM)
- B1515 Raloxifene HCl中文名: 盐酸雷洛昔芬Target: Estrogen and Related ReceptorsSummary: 雌激素受体(ER)调节剂
- B5421 (Z)-4-Hydroxytamoxifen中文名: 4-羟基他莫昔芬Target: Estrogen and Related ReceptorsSummary: 雌激素受体(ER)调节剂