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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- A4064 NVP-BEP800Target: HSP90Summary: 全合成的HSP90β口服抑制剂
- A4061 IPI-504 (Retaspimycin hydrochloride)3 Citation中文名: 瑞他霉素盐酸盐Target: HSP90Summary: Hsp90抑制剂
- B7393 GeduninTarget: HSP90Summary: 天然的Hsp90抑制剂
- A4056 AT13387Target: HSP90Summary: Hsp90抑制剂
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- N1359 Magnolol中文名: 厚朴酚Target: CB1 Receptors|NO Donors / Precursors|CB2 ReceptorsSummary: NO/TNF-α产生的抑制剂;抗真菌剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- B1115 BAY 87-2243Target: Hypoxia Inducible Factors (HIFs)Summary: 有效的HIF-1选择性抑制剂