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- A1910 Bromodomain Inhibitor, (+)-JQ138 CitationTarget: BromodomainsSummary: BET bromodomain抑制剂。
- A3967 Lapatinib Ditosylate中文名: 二苯磺酸拉帕替尼Target: EGFR|ErbB-2Summary: EGFR / HER2抑制剂
- A8322 Neratinib (HKI-272)1 Citation中文名: 来那替尼Target: EGFRSummary: HER2/EGFR抑制剂
- A8324 LDN-193189Target: BMP and Other Activin ReceptorsSummary: ALK抑制剂
- A8555 Vandetanib (ZD6474)中文名: 凡德他尼Target: VEGFR|EGFRSummary: VEGFR2/EGFR拮抗剂
- A8357 AG-1478中文名: 酪氨酸磷酸化抑制剂 AG-1478Target: EGFRSummary: EGFR抑制剂
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: 有效的EGFR抑制剂
- B1438 BMS-794833Target: MET|Flk-1Summary: Met/VEGFR2抑制剂
- B3688 ML347Target: BMP and Other Activin ReceptorsSummary: 有效的BMP受体选择性抑制剂
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂