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- A8322 Neratinib (HKI-272)1 Citation中文名: 来那替尼Target: EGFRSummary: HER2/EGFR抑制剂
- A8555 Vandetanib (ZD6474)中文名: 凡德他尼Target: VEGFR|EGFRSummary: VEGFR2/EGFR拮抗剂
- A8357 AG-1478中文名: 酪氨酸磷酸化抑制剂 AG-1478Target: EGFRSummary: EGFR抑制剂
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: 有效的EGFR抑制剂
- A2574 Aprotinin1 Citation中文名: 抑酶肽Target: Trypsin|Chymotrypsin|Kallikrein|TrypsinogenSummary: 牛胰蛋白酶抑制剂
- B6962 CMPD-1Target: Microtubules/Tubulins|MK2Summary: p38α介导的MK2a磷酸化的抑制剂
- A8435 Furosemide中文名: 呋塞米Target: Na /K /Cl- Symporters (NKCCs)|GABAA ReceptorsSummary: GABAA受体拮抗剂
- C5545 MK2 Inhibitor IVTarget: MK2Summary: 高选择性、非ATP竞争性MK2抑制剂
- A3320 CO-1686 (AVL-301)1 CitationTarget: EGFRSummary: EGFR抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂