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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- A8351 VX-809中文名: 鲁玛卡托Target: CFTRSummary: CFTR调节剂
- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- B3225 BAF312 (Siponimod)1 Citation中文名: 辛波莫德Target: S1P receptorsSummary: S1P受体激动剂
- B7634 RP 001 hydrochlorideTarget: S1P receptorsSummary: S1P1受体激动剂
- A8548 Fingolimod (FTY720)中文名: 盐酸芬戈莫德Target: S1P receptorsSummary: S1P受体激动剂
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- A2664 VX-661Target: CFTRSummary: F508del CFTR校正子
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂