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- N1659 1-Deoxynojirimycin中文名: 1-脱氧野尻霉素Target: GlucosidasesSummary: anti-cancer medicine
- A4377 Evacetrapib (LY2484595)Target: CETPSummary: 强效的CETP选择性抑制剂
- A4375 Anacetrapib (MK-0859)1 Citation中文名: 安塞曲匹Target: CETPSummary: RhCETP/突变型 CETP(C13S) 抑制剂
- B7785 LDN 209929 dihydrochlorideTarget: haspin kinaseSummary: Haspin激酶抑制剂