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- A1910 Bromodomain Inhibitor, (+)-JQ138 CitationTarget: BromodomainsSummary: BET bromodomain抑制剂。
- B7590 Quinidine中文名: 奎尼丁Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)Summary: 降低Na+和K+通道电流
- B6674 Anisomycin中文名: 茴香霉素Target: p38|JNK|SAPKSummary: JNK激动剂
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂
- A8513 Riluzole中文名: 力鲁唑Target: Voltage-gated Sodium (NaV) Channels|glutamate releaseSummary: 钠通道抑制剂
- B1013 GSK1324726ATarget: BromodomainsSummary: BET蛋白抑制剂
- B2272 Phenytoin sodium中文名: 苯妥英钠Target: Voltage-gated Sodium (NaV) ChannelsSummary: 钠通道稳定剂
- B2274 Proparacaine HCl中文名: 盐酸丙美卡因Target: Voltage-gated Sodium (NaV) ChannelsSummary: 电压门控钠通道拮抗剂
- B1420 Bupivacaine HCl中文名: 盐酸布比卡因Target: Voltage-gated Sodium (NaV) ChannelsSummary: 麻醉药
- A8181 (-)-JQ14 CitationTarget: BromodomainsSummary: (+)-JQ1的立体异构体,可作为阴性对照物。