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- A4071 Fluorouracil (Adrucil)3 Citation中文名: 氟尿嘧啶Target: Thymidylate SynthaseSummary: 胸苷酸合成酶抑制剂,抗肿瘤药物。
- A4429 Vialinin ATarget: Deubiquitinating enzymes (DUBs)|IL Receptors|CCL2Summary: USP/IsoT/UCH-L1 DUB抑制剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- A3708 Pentostatin1 Citation中文名: 喷司他丁Target: Adenosine DeaminasesSummary: 腺苷脱氨酶抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂