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- A3885 TozadenantTarget: Adenosine A2A ReceptorsSummary: 腺苷2A受体拮抗剂
- A3735 PreladenantTarget: Adenosine A2A ReceptorsSummary: 腺苷A2A受体拮抗剂
- A8454 Istradefylline (KW-6002)中文名: 伊曲茶碱Target: Adenosine A2A ReceptorsSummary: 选择性A2A受体拮抗剂
- A1932 (-)-Huperzine A中文名: 石杉碱甲Target: NMDA Receptors|AChESummary: NMDA受体拮抗剂/AChE抑制剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂